Products

Active Pharmaceutical Ingredient Version: 202303

No.Product nameCAS numberRemarks
1,Entecavir Monohydrate恩替卡韦209216-23-9USDMF25200
R1-CEP 2016-152 –Rev 00
CADMF 2013-061 JP 227MF10302 TW DMF(64)0702
Y20170000439
2,Pranlukast
普仑司特
150821-03-7JP 228MF10119
3,Miglitol
米格列醇
72432-03-2JP 228MF10052
Y20170001242
4,Febuxostat
非布司他
144060-53-7(Form G) USDMF 29716 (Form G) CADMF2016-190
(Form G)ASMF Approved
(Form A)EMEA/ASMF/ 01386
(Form A)Y20190000927
5,Posaconazole
泊沙康唑
171228-49-2ASMF Approved USDMF29731
Y20180001585
6,Ticagrelor
替格瑞洛
274693-27-5EU/ASMF/00236
R0-CEP 2021-081-Rev 00
7,Apixaban
阿哌沙班
503612-47-3USDMF EU/ASMF/00292 CADMF 2018-151
8,Nebivolol Hydrochloride盐酸奈必洛尔152520-56-4ASMF Approved USDMF 29730
R0-CEP 2022-170-Rev 00
Y20230000174
9,Macitentan
马昔腾坦
441798-33-0ASMF Available USDMF Y20220001020
No.Product nameCAS numberRemarks
10,Efinaconazole
艾氟康唑
164650-44-6ASMF USDMF 32076
CADMF 2019-133 JP 305MF10025
11,Tasimelteon
他司美琼
609799-22-6USDMF 32077
12,Ramelteon
雷美替胺
196597-26-9USDMF 33719 JP 303MF10095 TW DMF(64)4208
13,Sugammadex Sodium
舒更葡糖钠
343306-79-6USDMF 35151 Y20200000429 EU/ASMF/00463
14,Tofacitinib citrate
枸橼酸托法替布
540737-29-9USDMF 35152 Y20210000144
15,Sitafloxacin Hydrate 西他沙星163253-35-8JP 228MF10177 Y20200000899
16,Calcium Saccharate
葡萄糖二酸钙
5793-89-5F20200000453
17,Asenapine
阿塞那平
65576-45-6DMF 2024.Q1
    
18,Pilocarpine Hydrochloride 盐酸毛果芸香碱54-71-7USDMF 038901
CEP application submitted
19,Isavuconazonium Sulfate
艾沙康唑硫酸盐
946075-13-4DMF: 2024 Q2
20,Repirinast
瑞吡司特
73080-51-0DMF: 2024 Q2
21,Lumateperone Tosylate
对甲苯磺酸芦玛哌酮
1187020-80-9DMF: 2024 Q1
22,Dapagliflozin
达格列净
461432-26-8DMF: 2024 Q2
23,Empagliflozin
依帕列净
864070-44-0DMF: 2024 Q3
24,Lifitegrast
立他司特
1025967-78-5DMF:2024 Q2
25,Avatrombopag
阿伐曲泊帕
570406-98-3DMF: 2024 Q1
26,Eliglustat
依鲁司他
491833-29-5ASMF ready (Tartrate)
No.Product nameCAS numberRemarks
27,Azvudine
阿兹夫定
1011529-10-4Y20230000006
28,Sapropterin
沙丙蝶呤
62989-33-7R&D
29,D(-)-Penicillamine
青霉胺
52-67-5R&D
30,Galanthamine
加兰他敏
357-70-0R&D
31,Rimegepant
瑞美吉泮
1289023-67-1R&D
32,Enzalutamide
恩杂鲁胺
915087-33-1R&D
33,Eflornithine HCl
盐酸依氟鸟氨酸
68278-23-9R&D
34,Diquafosol sodium
地夸磷索四钠
211427-08-6R&D
35,Bedaquiline
富马酸贝达喹啉
845533-86-0R&D
No.Product nameCAS numberRemarks
36,Roxadustat
罗沙司他
808118-40-3R&D
37,Deferasirox
地拉罗司
201530-41-8R&D
38,Relugolix
瑞卢戈利
737789-87-6R&D
39,Elagolix sodium
噁拉戈利钠
832720-36-2R&D
40,Taltirelin
他替瑞林
103300-74-9R&D
41,Teprenone
替普瑞酮
6809-52-5R&D
42,Nalfurafine HCl
盐酸纳呋拉啡
152658-17-8R&D
43,Carbidopa and Levodopa
卡左双多巴
28860-95-9
& 59-92-7
R&D
No.Product nameCAS numberRemarks
44,Imatinib mesilate
甲磺酸伊马替尼
220127-57-1EU/ASMF/00669
45,Cabozantinib
卡博替尼
849217-68-1DMF: 2024 Q2
46,Ruxolitinib (Phosphate)
(磷酸)芦可替尼
941678-49-5
& 1092939-17-7
DMF: 2024 Q1
47,Palbociclib
哌柏西利
571190-30-2DMF: 2023 Q4
48,Lenvatinib mesilate
甲磺酸仑伐替尼
857890-39-2DMF: 2023 Q4
49,Olaparib
奥拉帕尼
763113-22-0DMF: 2024 Q2
No.Product nameCAS numberRemarks
50,Trametinib dimethyl sulfoxide曲美替尼二甲亚砜1187431-43-1DMF: 2024 Q3
51,Dabrafenib mesilate
甲磺酸达拉非尼
1195768-06-9DMF: 2024 Q3
52,Osimertinib mesilate 奥西替尼1421373-66-1DMF: 2024 Q4
53,Nilotinib
尼洛替尼
641571-10-0R&D
54,Upadacitinib
乌帕替尼
1310726-60-3R&D
55,Pacritinib
帕克替尼
937272-79-2R&D
No.Product nameCAS numberRemarks
56,Homoharringtonine
高三尖杉酯碱
26833-87-4R&D
57,Harringtonin
三尖杉酯碱
26833-85-2R&D
58,6-Mercaptopurine 6-巯基鸟嘌呤154-42-7R&D
59,5-Azacytidine
阿扎胞苷
320-67-2R&D
60,Plerixafor
普乐沙福
110078-46-1R&D
61,Ixazomib
伊沙佐米
1201902-80-8R&D
62,Arotinolol Hydrochloride盐酸阿罗洛尔101540-26-5R&D
No.Product nameCAS numberRemarks
63,Vildagliptin
维达列汀
274901-16-5R&D
64,Cangrelor
坎格雷洛
163706-06-7R&D
65,Apremilast
阿普斯特
608141-41-9R&D
66,Betrixaban
贝曲西班
330942-05-7R&D
67,Lesinurad
来司诺雷
878672-00-5R&D
68,Brexpiprazole
依匹唑派
913611-97-9R&D
69,Remogliflozin329045-45-6R&D
70,Crisaborole
克立硼罗
906673-24-3R&D
71,Selexipag
赛乐西帕
475086-01-2R&D
No.Product nameCAS numberRemarks
72,Ravuconazole
拉夫康唑
182760-06-1R&D
73,Rotigotine
罗替戈汀
99755-59-6R&D
74,Elvitegravir
埃替格韦
697761-98-1R&D
75,Riociguat
利奥西呱
625115-55-1R&D
76,Zafirlukast
扎鲁司特
107753-78-6R&D
77,Istradefylline
伊曲茶碱
155270-99-8R&D
78,Miglustat
米格鲁特
72599-27-0R&D
79,Migalastat108147-54-2R&D
80,Edoxaban
依度沙班
480449-70-5R&D
No.Product nameCAS numberRemarks
81,Atropine
阿托品
51-55-8R&D
82,Scopolamine
东莨菪碱
51-34-3R&D
83,Methylscopolamine Bromide
甲溴东莨菪碱
155-41-9R&D
84,Scopolamine Butylbromide溴丁东莨菪碱149-64-4R&D
85,Scopolamine Hydrobromide 氢溴酸东莨菪碱114-49-8R&D
86,Oxitropium Bromide 氧托溴铵30286-75-0R&D
87,Ipratropium Bromide
异丙托溴铵
22254-24-6R&D
88,Flutropium bromide 氟托溴胺63516-07-4R&D
89,Aclidinium bromide  阿地溴铵320346-78-9R&D
No.Product nameCAS numberRemarks
90,Calcitriol
骨化三醇
32222-06-3R&D
91,Maxacalcitol
马沙骨化醇
103909-75-7R&D
92,Paricalcitol
帕立骨化醇
131918-61-1R&D
93,Alfacalcidol
阿法骨化醇
41294-56-8R&D
94,Doxercalciferol
度骨化醇
54573-75-0R&D
95,Calcifediol
骨化二醇
63283-36-3R&D
96,Tacalcitol
他卡西醇
57333-96-7R&D
No.Product nameCAS numberRemarks
97,Lubiprostone
鲁比前列酮
333963-40-9USDMF 30802
98,Latanoprost
拉坦前列腺素
130209-82-4CEP application submitted
99,Latanoprostene bunod
拉坦衍生物
860005-21-6DMF 2024.Q2
100,Tafluprost
他氟前列素
209860-87-7Y20220000747
101,Bimatoprost
比马前列素
155206-00-1DMF 2024.Q2
102,Travoprost
曲沃前列素
157283-68-6DMF 2023.Q4
103,Beraprost sodium
贝前列素
88475-69-8
88430-50-6
(acid)
R&D
104,Limaprost
利马前列素
74397-12-9R&D
105,Treprostinil sodium
曲前列素
289480-64-4
81846-19-7
(acid)
R&D
106,Misoprostol
米索前列醇
59122-46-2R&D
No.Product nameCAS numberRemarks
107,Isopropyl Unoprostone
乌诺前列酮异丙酯
120373-24-2R&D
108,Iloprost
伊洛前列素
78919-13-8R&D
109,Alprostadil (ProstaglandinE1)前列地尔(前列腺素 E1)745-65-3R&D
110,Dinoprostone (Prostaglandin E2)地诺前列酮 (前列腺
素 E2)
363-24-6R&D
111,Tiaprost
噻前列素
71116-82-0R&D
112,Dinoprost tromethamine
地诺前列素氨丁
三醇
38562-01-5
(Dinoprost 551-11-1)
R&D
113,Epoprostenol sodium
依前列醇钠
61849-14-7R&D
No.Product nameCAS numberRemarks
114,Carboprost Tromethamine 卡前列素氨丁三醇58551-69-2R&D
115,Etiproston
依替前列通
59619-81-7R&D
116,D-Cloprostenol Sodium
D-氯前列烯醇钠
62561-03-9R&D
117,D-Cloprostenol D-氯前列烯醇54276-22-1R&D
118,Trifluoromethyl Dechloro Ethylcloprostenola mide1005193-64-5R&D

Remark: Patented products available for research and development use ONLY as permitted under CFR 35
see 271 (e) (1). 

公司地址: 浙江省化学原料药基地临海园区东海第四大道5 号
Add: No.5, Donghai 4th Avenue, Zhejiang Chemical Materials Base Linhai Zone, Zhejiang, China
电话(Tel): +86-576-85589335 传真(Fax):+86-576-85589168
电子信箱(E-mail): sales@ausunpharm.com Website: http://www.ausunpharm.com

Intermediates

1.
.
(-)COD
(-)-Corey Lactone Diol Purity: ≥99.0 %
32233-40-2Prostaglandin Intermediates
2,BCOD
(-)-Corey Lactone Benzoate Purity: ≥99.0 %
39746-00-4
3,BPCOD
(-)-Corey Lactone p-Phenyl Benzoate Purity: ≥99.0 %
31752-99-5
4,TPPB
(4-carboxybutyl)triphenylphosphonium bromide
Purity: ≥99.0 %
17814-85-6
5,BMP
Dimethyl(2-oxo-4-phenylbutyl)phosphonate Purity: ≥94.0 %
41162-19-0Bimatoprost & Latanoprost Intermediates
6,BP-2
(3aR,4R,5R,6aS)-Hexahydro-5-hydroxy-4- [(1E,3R)-3-hydroxy-5-phenyl-1-pentenyl]-2H- cyclopenta[b]furan-2-one
Purity: ≥99.0 %
41639-74-1
7,LT-DI
(3aR,4R,5R,6aS)-Hexahydro-5-hydroxy-4- [(3R)-3-hydroxy-5-phenylpentyl]-2H- cyclopenta[b]furan-2-one
Purity: ≥99.0 %
145667-75-0
8,TVP
Dimethyl[2-Oxo-3-(3-trifluoromethyl- phenoxy)-propyl]phosphonate
Purity: ≥93.0 %
54094-19-8Travoprost Intermediates
9,TV-DI
(3aR,4R,5R,6aS)-Hexahydro-5- hydroxy-4-39-[(1E,3R)-3-hydroxy-4-(3- trifluoromethyl)phenoxy-1-butenyl]-2H- cyclopenta[b]furan-2-one
Purity: ≥99.0 %
53872-60-9
10,ETP
Dimethyl (3-phenoxy-2-oxopropyl) phosphonate
Purity: ≥95.0 %
40665-68-7Tafluprost Intermediates
11,TF-BF
(3aR,4R,5R,6aS)-5-(benzoyloxy)-4-[(1E)-  3,3-
difluoro-4-phenoxy-1-buten-1-yl] hexahydro-2H-Cyclopenta[b]furan-2-one
Purity: ≥99.0 %
209861-00-7
12,Diethyl(3-pyridyl)borane Purity≥99.0%89878-14-8Abiraterone intermediate
13,4,4-difluorocyclohexylcarboxylic acid122665-97-8Maraviroc Intermediate
14,F-TEDA-BF4 (Selectfluor)
Purity≥96.0%
140681-55-6 
15,苄基DBU 氯化物
Benzyl-DBU-Chloride
49663-94-7 

Remark: Patented products available for research and development use ONLY as permitted under CFR 35
see 271 (e) (1).

公司地址: 浙江省化学原料药基地临海园区东海第四大道5 号
Add: No.5, Donghai 4th Avenue, Zhejiang Chemical Materials Base Linhai Zone, Zhejiang, China
电话(Tel): +86-576-85589335 传真(Fax):+86-576-85589168
电子信箱(E-mail): sales@ausunpharm.com Website: http://www.ausunpharm.com